Ethylflualprazolam, Ethylmidazolam & Cycloproflualprazolam?

[kemdawg99]

I see all 3 popping up on Reddit & the onions (source is from an odd SE Asian country lol)

Anyone know of a domestic vendor or Chinese offering it yet? Im sure they'll make their way over here

Or any guinea pigs reading their magazines?

 

[LurkyLou]

Curious as well

 

[tiquanunderwood]

I've seen 3thylflu@lpr@z0lam for about 2-3 weeks now. I'm tempted since there's some domestic.



But I'm tapering so it'd probably be wise not to buy super tolerant b3nzos. But, I've done some researching in the scientific literature. Here's what I came up with thus far, I'll dive in deeper later, long day today.



"3thylflu@lpr@zol@m functions as a positive allosteric modulator of the GABA-A receptor. It binds to specific sites on the receptor complex, distinct from where the primary neurotransmitter gamma-aminobutyric acid (GABA) binds, which in turn enhances the frequency of chloride ion channel opening when GABA is present. This increased chloride influx hyperpolarizes the neuron membrane, making it less excitable and reducing overall neural signaling in the central nervous system."

So that's how these compounds function. Some bind to more sites than others, therefore causing the G@b@ A neurotransmitter to open and allow a more intense effect. I could be wrong. But different effects and sometimes more intense withdrawal symptoms happen after only a short use with some of these. Like cl0br0, which I'm pretty sure smashes most of the sites leaving the G@BA A transmitter to shut off/open and let the ch3m do its magic.

^^I assume that's why different b3nz0s have different qualities. Sometimes not majorly, but for example, there's some for insomnia and severe sleep issues, commonly called hypnotics (m1d@z0l@m, n1tr@z3p@m, etc.), some for panic disorder (@lpr@z0l@m and cl0n@z3p@m are the 2 in the states that are approved for this treatment), and then there's the Generalized Anxiety Disorder and muscle relaxation b3nz0$ (the gold standard for this is v@l1um). If you have a doc, in the states they'd probably start you on @t1v@n, if they give you a BZD, but I'm not a big fan of its shorter half life. It does do its job though, which these days is primarily in detox and treatment centers, alongside l1br1ium and v@l1um. But it's still commonly prescribed, just gotta take it twice per day at least without googling the half life. I know most of them but @t1v@n I can take or leave so I didn't memorize that one. It does its job, just nothing special or specific like some of the BZDs have.

Sorry got off topic. So, it turns out this is another BZD that China synthed that is a partial agonist of the G@B@ A receptor, br0m0n0rd1@z3p@m. Therefore, in theory there should be a ceiling dose, kind of like how sub0x0ne works. Actually, br0m0nor is also a partial agonist of G@BA A and I can tell I feel a lot better on that for a regular med, than lets say cl0bro or br0m@z. Hated the rebound anxiety. They just saturate the receptor and its subtypes so heavily. I find the withdrawal much worse as well. I know v@l1ium is a full agonist, but it's pretty mild, has a long half life, and it's pretty effective for short term GAD. I wouldn't use any of these long term (but look who's talking). But, I believe br0m0n0r could have a ceiling effect. And it definitely does not hit the near amount of receptor sites as the very potent ones.

I've been in the game for awhile, so please don't take this as advice, I'm just trying to provide my 2 cents and educate someone, anyone.



Anyways, when I come with more, I'll be back. Only had time to type about this one. There's not a lot out there.

That's it. Thanks!